@article{319c9e8b01a6418885c18b89ea1f301e,
title = "Acyclic and cyclic thioenamino peptides: solution- and solid-phase synthesis",
abstract = "Seven- and 10-membered cyclic thioenamino peptides, that is, 1,4-thiazepinone (11) and cyclic thioenamino peptide 9 (which represents a potential γ-turn mimetic), were synthesized, and the structure of 11 was secured by X-ray diffraction analysis of its TFA salt. The aforementioned compounds were prepared in solution and by solid-phase synthesis. Additionally, we have prepared thioenamino diketopiperazine synthon 16.",
keywords = "Cyclic peptides, Endiamine, FGly, Solid-phase synthesis, Thioenamine",
author = "Lee Goren and Doron Pappo and Israel Goldberg and Yoel Kashman",
note = "Funding Information: We thank the Israeli Science Foundation for financial support, Grant \# 180/05, Dr. Amira Rudi for her help with NMR measurements, Dr. Moshe Portnoy for helpful discussions, Ms. Yael Kogon for her contribution to this project, and Dr. Ayelet Sacher (of the Maiman Institute for Proteome Research, Tel Aviv University) for performing the electrospray mass measurements. ",
year = "2009",
month = mar,
day = "4",
doi = "10.1016/j.tetlet.2008.12.072",
language = "אנגלית",
volume = "50",
pages = "1048--1050",
journal = "Tetrahedron Letters",
issn = "0040-4039",
publisher = "Elsevier Ltd.",
number = "9",
}